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MICRONEEDLE-ARRAY PATCHES WITH GLUCOSE-RESPONSIVE MATRIX FOR CLOSED-LOOP INSULIN DELIVERY
MICRONEEDLE-ARRAY PATCHES WITH GLUCOSE-RESPONSIVE MATRIX FOR CLOSED-LOOP INSULIN DELIVERY
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机译:微糖阵列与葡萄糖敏感矩阵的闭环胰岛素输送
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摘要
Disclosed are compositions and methods for microneedle patches comprising copolymer designed for glucose triggered insulin delivery. In one aspect, disclosed herein are microneedle patches comprising insulin loaded copolymers; wherein the insulin dissociates from the microneedle in an hyperglycemic environment; wherein the copolymer comprises poly(N-vinylpyrrolidone-co-2-(dimethylamino)ethyl acrylate-co-3-(acrylamido)phenylboronic acid and methods of their use.
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机译:公开了用于微针贴剂的组合物和方法,其包括设计用于葡萄糖触发的胰岛素递送的共聚物。一方面,本文公开了包含载有胰岛素的共聚物的微针贴剂。在高血糖环境中,胰岛素从微针上解离;其中共聚物包含聚( N I>-乙烯基吡咯烷酮- co </ I> -2-(二甲基氨基)乙基丙烯酸酯- co </ I> -3-(丙烯酰胺基)苯基硼酸及其使用方法。
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