Lewis Acid Catalyzed Reaction of Arylvinylidenecyclopropanes with Ethyl (Arylimino)acetates: A Facile Synthetic Protocol for Pyrrolidine and 1,2,3,4-Tetrahydroquinoline Derivatives

摘要

A number of pyrrolidine and 1,2,3,4-tetrahydroquinoline derivatives are prepared selectively in moderate to good yields by the reaction of arylvinylidenecyclopropanes 1 with ethyl (arylimino)acetates 2 in the presence of Lewis acid depending on the electronic nature both of 2 and R~1 or R~2 aromatic groups of 1.