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机译:通过合成8-烷氧基噻吩并2,3-c异喹啉-5(4H)-酮的PARP抑制剂TIQ-A衍生物
Faculty of Biochemistry and Molecular Medicine &;
Biocenter Oulu, University of Oulu;
Research Unit of Sustainable Chemistry, University of Oulu;
Drug &;
Target Discovery, Department of Pharmacy &;
Pharmacology, University of Bath;
机译:A novel Syk family kinase inhibitor: design, synthesis, and structure-activity relationship of 1,2,4-triazolo(4,3-c)pyrimidine and 1,2,4-triazolo(1,5-c)pyrimidine derivatives.
机译:Synthesis and evaluation of 2‐(4‐4‐acetylpiperazine‐1‐carbonyl phenyl)‐1H‐benzodimidazole‐4‐carboxamide derivatives as potential PARP‐1 inhibitors and preliminary study on structure‐activity relationship
机译:Discovery of Quinazoline-2,4(1H,3H)-dione Derivatives Containing 3-Substituted Piperizines as Potent PARP-1/2 Inhibitors-Design, Synthesis, In Vivo Antitumor Activity, and X-ray Crystal Structure Analysis
机译:PARP抑制剂TIQ-A的衍生物8-烷硫基23-c异喹啉-5(4H)-ones的合成
机译:In silico Identification of structure Requirement for Novel Thiazole and Oxazole Derivatives as potent Fructose 1,6-Bisphosphatase Inhibitors