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机译:发现新的Celastrol衍生品作为HSP90-CDC37互动破坏者,具有抗肿瘤活动
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
China Pharmaceut Univ Sch Tradit Chinese Pharm Dept Nat Med Chem State Key Lab Nat Med 24 Tong Jia Xiang Nanjing 210009 Jiangsu Peoples R China;
机译:发现新的Celastrol衍生品作为HSP90-CDC37互动破坏者,具有抗肿瘤活动
机译:作为HSP90-CDC37相互作用的氨基苯并噻唑衍生物发现18β-甘草酸共轭氨基苯噻唑衍生物,其抑制细胞迁移和逆向耐药性
机译:新型HSP90抑制剂DCZ3112通过破坏HSP90-CDC37相互作用来施加抗HER2阳性乳腺癌的有效抗肿瘤活性
机译:硝基唑类抗肿瘤活性的定量结构活性关系(QSAR):母体化合物及其硝基苯醌自由基和亚硝基苯醌自由基衍生物的比较分析
机译:发现具有有效的抗增殖和抗肿瘤活性的小分子二氢喹啉酮抑制剂会导致灾难性的细胞分裂。
机译:在计算机上发现了小分子Ras抑制剂这些抑制剂通过阻断Ras与效应子的相互作用而显示出抗肿瘤活性
机译:发现新的Celastrol衍生品作为HSP90CDC37互动破坏者,抗肿瘤活动