...
机译:一种新的大鼠衍生物,N-(4-(羟基氨基甲酰基)苄基)-1-(4-甲氧基苯基)-9H-吡啶[3,4-B]吲哚-3-甲酰胺(HBC),作为组蛋白脱乙酰酶抑制剂:体外 抗溶解,细胞凋亡诱导,细胞周期骤停和抗致锑效应
Nantong Univ Affiliated Hosp Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Sch Pharm Nantong 226001 Peoples R China;
Nantong Univ Affiliated Hosp Nantong 226001 Peoples R China;
Nantong Univ Affiliated Hosp Nantong 226001 Peoples R China;
Nantong Univ Affiliated Hosp Nantong 226001 Peoples R China;
Harmine derivative; Antitumor activity; Histone deacetylase inhibitor; Apoptosis; Cell cycle arrest; Antimetastatic activity;
机译:一种新的大鼠衍生物,N-(4-(羟基氨基甲酰基)苄基)-1-(4-甲氧基苯基)-9H-吡啶[3,4-B]吲哚-3-甲酰胺(HBC),作为组蛋白脱乙酰酶抑制剂:体外 抗溶解,细胞凋亡诱导,细胞周期骤停和抗致锑效应
机译:在非小细胞肺癌(NSCLC)细胞中,组蛋白脱乙酰基酶抑制剂曲古抑菌素A对伽马辐射诱导的细胞周期停滞和凋亡的敏感性。
机译:组蛋白脱乙酰基酶抑制剂曲古他汀A对EBV转化的B淋巴母细胞的细胞周期阻滞和裂解诱导作用。
机译:介导细胞毒性药物,组蛋白脱乙酰基酶抑制剂或血清剥夺的细胞周期停滞或凋亡的介导者。
机译:新型组蛋白脱乙酰化酶抑制剂AR-42抑制GP130 / Stat3途径并在多个骨髓瘤细胞中诱导细胞凋亡和细胞周期停滞
机译:新型组蛋白脱乙酰基酶抑制剂AR-42抑制gp130 / Stat3途径并诱导多发性骨髓瘤细胞凋亡和细胞周期停滞