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机译:1-(1H-吲哚-1-基)乙酮衍生物的发现和优化作为CBP / EP300溴阳瘤抑制剂,用于治疗抗阉割前列腺癌
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Univ Chinese Acad Sci 19 Yuquan Rd Beijing 100049 Peoples R China;
Jilin Univ Sch Pharmaceut Sci 1266 Fujin Rd Changchun 130021 Jilin Peoples R China;
Univ Auckland Auckland Canc Soc Res Ctr Sch Med Sci Private Bag 92019 Auckland New Zealand;
Univ Auckland Auckland Canc Soc Res Ctr Sch Med Sci Private Bag 92019 Auckland New Zealand;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
Jinan Univ Sch Pharm 601 Huangpu Ave West Guangzhou 510632 Guangdong Peoples R China;
Guangzhou Med Univ Guangdong Prov Key Lab Biocomp Joint Sch Life Sci Chinese Acad Sci Guangzhou;
CBP; EP300; Prostate cancer; Bromodomain inhibitor;
机译:1-(1H-吲哚-1-基)乙酮衍生物的发现和优化作为CBP / EP300溴阳瘤抑制剂,用于治疗抗阉割前列腺癌
机译:基于结构的发现和优化苯并[ D i>]异恶唑衍生物作为有效和选择性的BET抑制剂,用于抵抗抗阉割前列腺癌(CRPC)
机译:含苯并嗪酮的3,5-二甲基异恶唑衍生物作为β溴抑制剂,用于治疗抗阉割前列腺癌
机译:转移激素敏感和阉割的前列腺癌:进步和持续发现的十年
机译:测定用于去势抵抗性前列腺癌的治疗剂的新代谢产物。
机译:Y08197是一种新颖和选择性CBP / EP300溴琼肿瘤抑制剂用于治疗前列腺癌
机译:基于片段的选择性和细胞活性苯并二氮醌CBP / EP300 Bromodomain抑制剂的发现(CPI-637)