CAS Key Laboratory of Receptor Research;
CAS Center for Excellence in Molecular Cell Science;
Center for Biotherapeutics Discovery Research;
Shanghai Institute of Materia Medica Chinese Academy of Sciences;
Shanghai 201203;
China;
School of Pharmaceutical Science and Technology;
Hangzhou Institute of Advanced Study;
Hangzhou 310024;
China;
University of Chinese Academy of Sciences;
Beijing 100049;
China;
School of Chinese Materia Medica;
Nanjing University of Chinese Medicine;
Nanjing 210023;
China;
School of Life Science;
Liaocheng University;
Liaocheng 252059;
China;
Site-specific ADCs; ENGase; LacNAc; One-step assembly; Potent in vivo efficacy;