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CRYSTALLINE FORM OF HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

机译:结晶形式的杂环化合物,其制备方法及其应用

摘要

Provided are a crystalline form of a compound represented by formula A, the crystalline form being crystalline form I, crystalline form II, crystalline form III, crystalline form IV, crystalline form V, crystalline form VI, crystalline form VII, crystalline form VIII or crystalline form IX, a preparation method therefor, a composition thereof, and an application thereof in the preparation of a P2X3 receptor antagonist or an application thereof in the preparation of drugs preventing and/or treating pains, urinary tract illness or respiratory system illness. The compound has high P2X3 antagonist activity, and has good selectivity, low toxicity, good metabolic stability and little taste influence.
机译:是由式A表示的化合物的结晶形式,结晶形式是结晶形式I,结晶形式II,结晶形式III,结晶形式IV,结晶形式V,结晶形式VI,结晶形式VII,结晶形式VIII或结晶。 形成IX,其制备方法,其组合物及其应用在制备P2X3受体拮抗剂或其应用中,在制备药物中预防和/或治疗疼痛,泌尿道或呼吸系统疾病。 该化合物具有高p2x3拮抗剂活性,具有良好的选择性,低毒性,良好的代谢稳定性和味道少。

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