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Modified dextran complex containing lysine-urea-glutamate pharmacophore

机译:改性葡萄糖络合物含有赖氨酸 - 尿素 - 谷氨酸药物团

摘要

The present invention is related to modified dextran conjugates, such as guanidine-dextran conjugates, comprising a PSMA binding tripeptide. The present invention further discloses a method for preparation of said conjugates as well as their use. The conjugate of the present invention can be used for treating or diagnosis of a disease or a condition associated with expression of prostate specific membrane antigen (PSMA).
机译:本发明涉及修饰的葡聚糖缀合物,例如胍丁烷缀合物,其包含PSMA结合三肽。 本发明进一步公开了一种制备所述缀合物以及它们的使用方法。 本发明的缀合物可用于治疗或诊断疾病或与前列腺特异性膜抗原(PSMA)的表达相关的病症。

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