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CRYSTALLINE FORM OF FLUVATINIB OR FLUVATINIB METHANESULFONATE AND PREPARATION METHOD THEREFOR

机译:氟嘌呤或氟伐替尼甲烷磺酸盐的结晶形式和制备方法

摘要

A crystalline form of fluvatinib or fluvatinib methanesulfonate, and a preparation method therefor. The crystalline form I of the fluvatinib has characteristic diffraction peaks as shown in FIG. 1. The crystalline form of the fluvatinib methanesulfonate may take multiple forms, including seven crystalline forms, forms I-VII, wherein crystalline form III has characteristic diffraction peaks as shown in FIG. 9. Said crystalline forms are suited to manufacturing processes for fluvatinib methanesulfonate formulations.
机译:氟伐替尼或氟伐替尼甲烷磺酸盐的结晶形式,及其制备方法。 氟瓦替尼的结晶形式I具有特征性衍射峰,如图2所示。 1.氟伐替尼甲磺酸盐的结晶形式可以采用多种形式,包括七种晶体形式,形成I-VII,其中结晶形式III具有特征衍射峰,如图2所示。 9.所述结晶形式适用于氟伐替尼甲磺酸盐制剂的制造方法。

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