首页> 外国专利> CRYSTALLINE SOLVATES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL) METHYL) PHENYL)-D-GLUCITOL DERIVATIVES WITH ALCOHOLS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES

CRYSTALLINE SOLVATES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL) METHYL) PHENYL)-D-GLUCITOL DERIVATIVES WITH ALCOHOLS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES

机译:(1S)-1,5- Anydro-1-C-(3 - ((苯基)甲基)苯基)-D-葡糖酚衍生物的结晶溶剂化物作为醇作为SGLT2抑制剂用于治疗糖尿病

摘要

The present invention relates to a pharmaceutical composition comprising a therapeutically effective amount of a crystalline (2S,3R,4S,5S,6R)-2-[4-chloro-3-(4-ethoxy-benzyl)-phenyl] -6-hydroxymethyl-2-methoxy-tetrahydro-pyran-3,4,5-triol (S)-propylene glycol solvate (compound Ia) as SGLT2 inhibitor for treating diabetes.
机译:本发明涉及药物组合物,其包含治疗有效量的结晶量(2s,3r,4s,5s,6r)-2- [4-氯-3-(4-乙氧基 - 苄基) - 苯基] -6-羟甲基-2-甲氧基 - 四氢 - 吡喃-3,4,5-三醇 - 丙二醇溶剂化物(化合物IA)作为治疗糖尿病的SGLT2抑制剂。

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