首页> 外国专利> DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF HALLUCINATIONS ASSOCIATED WITH A NEURODEGENERATIVE DISEASE

DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF HALLUCINATIONS ASSOCIATED WITH A NEURODEGENERATIVE DISEASE

机译:亚芳基和芳基代芳亚芳基脲衍生物作为5-HT2A血清素受体的调节剂,可用于预防和治疗与神经变性疾病相关的幻觉

摘要

The present invention relates to certain pyrazole derivatives of Formula (I) and pharmaceutical compositions thereof that modulate the activity of the 5-HT2A serotonin receptor and their uses for the treatment and prophylaxis of visual hallucinations associated with Lewy Body dementia.
机译:本发明涉及一种式(I)和药物组合物的某种吡唑衍生物,其调节5-HT 2a-serotonin受体的活性及其用于治疗和预防与lewy的视觉幻觉的用途身体痴呆症。

著录项

  • 公开/公告号US2021177804A1

    专利类型

  • 公开/公告日2021-06-17

    原文格式PDF

  • 申请/专利权人 AXOVANT SCIENCES GMBH;

    申请/专利号US202017100528

  • 申请日2020-11-20

  • 分类号A61K31/415;A61K9/20;A61K45/06;A61K31/13;A61K31/135;A61K31/198;A61K31/27;A61K31/4045;A61K31/445;A61K31/55;A61K31/5513;A61K31/554;A61P25;

  • 国家 US

  • 入库时间 2022-08-24 19:24:45

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