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DUAL-TARGETED CARBONIC ANHYDRASE IX COMPLEX AND CONTRAST AGENT THEREOF

机译:双靶向碳酸酐酶IX复合物及其造影剂

摘要

Disclosed herein are a dual-targeted carbonic anhydrase IX complex, a contrast agent comprising the same, and a synthesizing method thereof. The dual-targeted carbonic anhydrase IX complex includes a carbonic anhydrase IX (CA9) binding peptide, a sulfonamide derivative, and a metal chelating agent. The dual-targeted carbonic anhydrase IX complex has potential for use as a molecular nuclear drug.
机译:本文公开了一种双靶向碳酸酐酶IX络合物,其造影剂是相同的,及其合成方法。双靶向碳酸酐酶IX配合物包括碳酸酐酶IX(CA9)结合肽,磺酰胺衍生物和金属螯合剂。双靶向碳酸酐酶IX复合物具有用作分子核药物的潜力。

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