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Methods for treating cancer with RORγ inhibitors

机译:用RORγ抑制剂治疗癌症的方法

摘要

The present invention provides compositions, methods, and kits comprising one or more RORγ inhibitors, alone or in combination with one or more anticancer drugs, such as an anti-androgen drug, that are useful for treating cancer, e.g., prostate cancer, such as castration-resistant prostate cancer (CRPC), and numerous other types of cancer including lung cancer, breast cancer, liver cancer, ovarian cancer, endometrial cancer, bladder cancer, colon cancer, lymphoma, and glioma.
机译:本发明提供了包含一种或多种RORγ抑制剂,单独或与一种或多种抗癌药物组合的组合物,方法和试剂盒,例如抗雄激素,可用于治疗癌症,例如前列腺癌,例如前列腺癌抗阉割的前列腺癌(CRPC),以及许多其他类型的癌症,包括肺癌,乳腺癌,肝癌,卵巢癌,子宫内膜癌,膀胱癌,结肠癌,淋巴瘤和胶质瘤。

著录项

  • 公开/公告号US10959984B2

    专利类型

  • 公开/公告日2021-03-30

    原文格式PDF

  • 申请/专利权人 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA;

    申请/专利号US201715701122

  • 发明设计人 HONGWU CHEN;JUNE X. ZOU;JUNJIAN WANG;

    申请日2017-09-11

  • 分类号A61K31/496;A61K31/167;A61K31/403;C07D209/56;C07D419/12;C07D401/12;C07D403/12;C07D405/12;C07K14/705;A61K31/18;A61K31/185;A61K31/4166;A61K31/4725;A61K31/655;A61K31/713;C12N15/113;

  • 国家 US

  • 入库时间 2022-08-24 17:58:48

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