首页> 外国专利> PROCESS FOR THE PREPARATION OF N- (METHOXYMETHYLEFPROCEDE FOR THE PREPARATION OF N- (METHOXYMETHYLFURYLMETHYLE) -6,7-BENZOMORPHANES-MORPHINANES URYLMETHYLE) -6,7-BENZOMORPHANES-MORPHINANES

PROCESS FOR THE PREPARATION OF N- (METHOXYMETHYLEFPROCEDE FOR THE PREPARATION OF N- (METHOXYMETHYLFURYLMETHYLE) -6,7-BENZOMORPHANES-MORPHINANES URYLMETHYLE) -6,7-BENZOMORPHANES-MORPHINANES

机译:制备N-(甲羟甲基方法的制备方法-6,7-苯甲硫基-吗啉的缩合戊烯基)-6,7-苯甲硫基-吗啡的制备法

摘要

Compound of the formula WHEREIN R1 and R2, which may be identical to or different from each other, are each hydrogen or alkyl of 1 to 3 carbon atoms, R3 is hydrogen or methyl, R4 is R5 is hydrogen, methyl or acetyl, AND NON-TOXIC, PHARMACOLOGICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF; THE COMPOUNDS AS WELL AS THEIR SALTS ARE USEFUL AS ANALGESICS.
机译:式中,R 1和R 2彼此相同或不同的化合物分别为氢或1-3个碳原子的烷基,R 3为氢或甲基,R 4为R 5为氢,甲基或乙酰基,并且有毒,药理学上可接受的酸加成盐;化合物及其盐可作为止痛药使用。

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