首页> 外国专利> ANTITUMORAL AGENTS, SUCH AS DAUNORUBICIN, HAVING AN IMPROVED ACTIVITY, OBTENTION THEREOF AND METHOD FOR ENHANCING THE ACTIVITY OF ANTITUMORAL AGENTS

ANTITUMORAL AGENTS, SUCH AS DAUNORUBICIN, HAVING AN IMPROVED ACTIVITY, OBTENTION THEREOF AND METHOD FOR ENHANCING THE ACTIVITY OF ANTITUMORAL AGENTS

机译:抗肿瘤活性剂,如柔红霉素,其活性得到改善,观察到其和增强抗微生物剂活性的方法

摘要

The antitumoral agent such as daunorubicin is brought in presence of a well determined quantity of a bifunctional bridging agent such as glutaraldehyde. The result is a form of a polymer product, which is unsoluble in an aqueous medium but which, when resuspended in an aqueous medium in the absence of glutaraldehyde, releases progressively the antitumoral agent in a soluble form, while preserving its antitumoral activity. Application: improvement of the treatment conditions by means of the antitumoral agents.
机译:在确定的双功能桥接剂(如戊二醛)存在的情况下,将抗肿瘤剂(如柔红霉素)带入。结果是聚合物产物的形式,其不溶于水性介质,但是当在没有戊二醛的情况下重悬于水性介质中时,以可溶形式逐渐释放抗肿瘤剂,同时保留其抗肿瘤活性。应用:通过抗肿瘤药改善治疗条件。

著录项

  • 公开/公告号WO8302946A1

    专利类型

  • 公开/公告日1983-09-01

    原文格式PDF

  • 申请/专利权人 INSTITUT PASTEUR;RELYVELD EDGAR HANS;

    申请/专利号WO1983FR00036

  • 发明设计人 RELYVELD EDGAR HANS;

    申请日1983-02-25

  • 分类号C07H15/24;A61K31/70;

  • 国家 WO

  • 入库时间 2022-08-22 10:36:15

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号