首页> 外国专利> Antibiotic derivatives, derived from cephalosporins with thiazolyl substituents, pharmaceutical preparations and salts thereof

Antibiotic derivatives, derived from cephalosporins with thiazolyl substituents, pharmaceutical preparations and salts thereof

机译:衍生自具有噻唑基取代基的头孢菌素的抗生素衍生物,药物制剂及其盐

摘要

The present invention relates to derivatives of the family of cephalosporins, of formula: ##STR1## in which ##STR2## is an acid, a salt or an ester of this acid, R.sub.1 is a group of form ##STR3## in which R. sub.A and R.sub.B are H or alkyl or form a saturated cyclobutyl or cyclopentyl ring and R.sub.C is H or COOH, R.sub.2 is a thiazolium salt or a OCOCH.sub.2 R.sub.D group in which R.sub.D is a 1,3-thiazol-4-yl group.PPThe invention also relates to a process for preparing the products of formula (I) and to drugs containing said products.
机译:本发明涉及头孢菌素家族的衍生物,其分子式为:其中,## STR2 ##是该酸的酸,盐或酯,R.sub.1是下列形式的基团:其中R A和R B是H或烷基或形成饱和的环丁基或环戊基环,R C是H或COOH,R 2是噻唑鎓盐或其中O D是1,3-噻唑-4-基的OCOCH 2 R D基团。P

本发明还涉及制备产物的方法。式(I)的化合物和含有所述产物的药物。

著录项

  • 公开/公告号US4476123A

    专利类型

  • 公开/公告日1984-10-09

    原文格式PDF

  • 申请/专利权人 SANOFI;

    申请/专利号US19820353890

  • 发明设计人 BERNARD LABEEUW;ALI SALHI;

    申请日1982-03-02

  • 分类号A61K31/545;C07D501/56;

  • 国家 US

  • 入库时间 2022-08-22 08:37:18

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号