Method for preparing Allyl Amine compounds as inhibitors of monoamine oxidase. Breakdown of Invention Patent 512.699 n

摘要

Method for preparing Allyl Amine compounds as inhibitors of monoamine oxidase.Comprising: (a) treating a compound of formula (iii) or (iv) with benzaldehyde in the presence of a Lower alcohol (Ethanol), to form Schiff base; b) treating the Schiff base with tetrafluoruroborato of trietiloxonio, to obtain an intermediate compound; and (c) HYDROLYZE The Compound. Rmedio to produce Allyl Amine oxidase inhibitors monoamine compounds of formula (i) or (ii).Where: R, dioxofenilo phenyl 3,4 - methylene -, 1 - or 2 - naphthyl and others; R1, c h, alkyl of 1 to 8 and others; X and y are mutually Independent, h, F, cl or BR, a radical of formula (V); R2, h Methyl or Ethyl, and Independent; IF m and N are integers between 0 to 4 h, being useful 4.se MBN Fly to the treatment of Psychiatric Disorders (Depression).