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seen framstella deaminoderivat of kallikrein and trypsin inhibitor from notorgan

机译:观察到来自诺加丹的激肽释放酶的弗拉姆氏菌脱氨基衍生物和胰蛋白酶抑制剂

摘要

A demaino kallikrein-trypsin inhibitor obtained from cattle organs is characterized by (a) 0 to 3 lysine residues and/or 3 to 6 arginine residues and/or 1 to 4 tyrosine residues; (b) the 10- and/or 21-tyrosine residues being unsubstituted or substituted by at least one nitro, nitroso or amino in the ortho position relative to the phenolic hydroxy group; and (c) having protease inhibitory activity of BPTI and elastase inhibition activity.
机译:从牛器官获得的去氢激肽释放酶-胰蛋白酶抑制剂的特征在于:(a)0至3个赖氨酸残基和/或3至6个精氨酸残基和/或1至4个酪氨酸残基; (b)10-和/或21-酪氨酸残基未被取代或在相对于酚羟基的邻位被至少一个硝基,亚硝基或氨基取代; (c)具有BPTI的蛋白酶抑制活性和弹性蛋白酶抑制活性。

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