首页> 外国专利> PROCESS FOR THE PREPARATION OF NOVEL DERIVATIVES OF 5-H PYRIDO 3 ', 4': 4,5 PYRROLO 3,2-C PYRIDINE WITH ANTITUMOR ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

PROCESS FOR THE PREPARATION OF NOVEL DERIVATIVES OF 5-H PYRIDO 3 ', 4': 4,5 PYRROLO 3,2-C PYRIDINE WITH ANTITUMOR ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

机译:具有反活性和包含相同成分的5-H吡咯烷酮<3',4':4,5>吡咯烷<3,2-C>吡啶的新型衍生物的制备方法

摘要

Derivatives of formula: IMAGE in which n denotes an integer from 2 to 4, R1 denotes hydrogen or a lower alkyl group, R2 and R3 denote hydrogen, a lower alkyl or hydroxyalkyl group and the tautomeric forms and addition salts with pharmaceutically acceptable inorganic or organic acids. Application in therapeutics.
机译:式:的衍生物,其中n表示2至4的整数,R1表示氢或低级烷基,R2和R3表示氢,低级烷基或羟烷基,并且互变异构形式和与药学上可接受的无机盐的加成盐或有机酸。在治疗中的应用。

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