首页> 外国专利> cis - or trans - 3.4 - the other ingredients are - n - 2 - (dimethylamino) - cyclopentyl - propioanilid and antidepressant with an n - (2 - aminocyclopentyl) - n - alkanoylanilid as active ingredient

cis - or trans - 3.4 - the other ingredients are - n - 2 - (dimethylamino) - cyclopentyl - propioanilid and antidepressant with an n - (2 - aminocyclopentyl) - n - alkanoylanilid as active ingredient

机译:顺式或反式3.4-其他成分为-正[2-(二甲基氨基)-环戊基]-丙苯胺和抗抑郁药,以正-(2-氨基环戊基)-正-烷酰基苯胺为有效成分

摘要

Novel N-(2-aminocyclopentyl)-N-alkanoyl anilides and 2-N-oxides thereof of the formula: IMAGE in which the substituents are defined in Claims 1 and 10, are prepared. These compounds are obtained by acylating N-(2-aminocyclopentyl)aniline on the nitrogen atom either with an anhydride of an organic carboxylic acid of the formula R-COOH or with a R-C (O)-chloride or R-C (O)-bromide. The corresponding N-oxides are prepared from these acylated compounds by oxidation with a percarbonic acid. The novel compounds which are obtained can be used as antidepressants.
机译:制备式:的新型N-(2-氨基环戊基)-N-链烷酰苯胺及其2-N-氧化物,其中取代基在权利要求1和10中定义。这些化合物通过用式R-COOH的有机羧酸的酸酐或R-C(O)-氯化物或R-C(O)-溴化物将氮原子上的N-(2-氨基环戊基)苯胺酰化而获得。由这些酰化的化合物通过用过碳酸氧化来制备相应的N-氧化物。所获得的新型化合物可以用作抗抑郁药。

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