首页> 外国专利> PROCESS FOR PREPARING SUBSTITUTED PYRIDO/1,2-C/IMIDAZO /1,2-A/BENZIMIDAZOLES AND PHARMACEUTICALS COMPRISING THE COMPOUNDS

PROCESS FOR PREPARING SUBSTITUTED PYRIDO/1,2-C/IMIDAZO /1,2-A/BENZIMIDAZOLES AND PHARMACEUTICALS COMPRISING THE COMPOUNDS

机译:制备取代的PYRIDO / 1,2-C /咪唑/ 1,2-A /苯并咪唑和包含该化合物的药物的方法

摘要

The invention relates to compounds of the formula IMAGE (I) in which R1 and R2 are identical or different and are hydrogen, alkyl, trifluoromethyl, halogen, alkoxycarbonyl, alkoxy or alkanoyl, R3, R4 and R5 are identical or different and are hydrogen, methyl, alkoxy or alkoxyethoxy, and R is hydrogen or a group SR6, in which R6 is the lone, unpaired electron of the 12-sulfenyl radical, hydrogen, optionally substituted alkyl, alkenyl, alkynyl, alkanoyl, optionally mono- or poly-substituted benzoyl, fuoryl, phenacyl, phenoxyacetyl, phenylacetyl or another conventional thiol-protective group, and to physiologically acceptable salts thereof, and to processes for their preparation, to their use as a gastric acid secretion inhibitor and to pharmaceutical preparations based on these compounds.
机译:本发明涉及式(I)的化合物,其中R1和R2相同或不同,并且为氢,烷基,三氟甲基,卤素,烷氧基羰基,烷氧基或烷酰基,R3,R4和R5相同或不同并且为氢,甲基,烷氧基或烷氧基乙氧基,且R为氢或SR6基团,其中R6为12-亚硫基基团的孤独,不成对的电子,氢,任选取代的烷基,烯基,炔基,炔基,任选单或多取代的苯甲酰基,氟甲酰基,苯甲酰基,苯氧基乙酰基,苯乙酰基或另一种常规的巯基保护基,及其生理上可接受的盐,及其制备方法,用作胃酸分泌抑制剂的用途以及基于这些化合物的药物制剂。

著录项

  • 公开/公告号HU194234B

    专利类型

  • 公开/公告日1988-01-28

    原文格式PDF

  • 申请/专利权人 HOECHST AGDE;

    申请/专利号HU19840003413

  • 申请日1984-09-10

  • 分类号C07D471/14;A61K31/395;

  • 国家 HU

  • 入库时间 2022-08-22 07:00:06

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