首页> 外国专利> COMPOUNDS POSSESSING BETA-ANTAGONISTIC AND ALPHA-ANTAGONISTIC PROERTIES, SUITABLE FOR LOWERING THE INTRAORBITAL PRESSURE, PHARMACEUTICAL COMPOSITION CONTAINING THESE COMPOUNDS, UTILIZATION THEREOF

COMPOUNDS POSSESSING BETA-ANTAGONISTIC AND ALPHA-ANTAGONISTIC PROERTIES, SUITABLE FOR LOWERING THE INTRAORBITAL PRESSURE, PHARMACEUTICAL COMPOSITION CONTAINING THESE COMPOUNDS, UTILIZATION THEREOF

机译:含有β-反义和α-反义性质的化合物,适合降低眶内压力,包含这些化合物的药物成分,并加以利用

摘要

The compounds having the formulae (I), (II), (III), (IV), (V), in which R is (VI), consist of a pattern derived from beta-blockers and an imidazolidine pattern possessing alpha-antagonistic properties. These compounds, which are new, therefore have the antagonistic properties of the beta-adreno-receptors and can consequently be used to lower the intraorbital pressure, in particular in glaucoma cases.
机译:其中R是(VI)的具有式(I),(II),(III),(IV),(V)的化合物由衍生自β-阻滞剂的图案和具有α-拮抗作用的咪唑烷图案组成属性。这些新的化合物因此具有β-​​肾上腺素受体的拮抗特性,因此可用于降低眼内压,特别是在青光眼病例中。

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