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2 * 44jikuroroo55furuorooansokukosanjudotai

机译:2 * 44九老郎55古郎Ansokuko-san柔道台

摘要

1. Claims (for the Contracting States : AT, BE, CH, DE, FR, GB, IT, LI, NL, SE) Cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-piperazino- quinoline-3-carboxylic acids of the formula I see diagramm : EP0078362,P10,F3 in which R denotes hydrogen, methyl, ethyl or beta-hydroxyethyl, and their pharmaceutically usable acid addition salts, alkali metal salts and hydrates, except 1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-piperazino- quinoline-3-carboxylic acid and its hydrochloride, 1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7- (4-methylpiperazino)-quinoline-3-carboxylic acid and 1-cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7- (4-ethylpiperazino)-quinoline-3-carboxylic acid hydroiodide. 1. Claims (for the Contracting State LU) 1-Cyclopropyl-6-fluoro-1,4-dihydro-4-oxo-7-piperazino- quinoline-3-carboxylic acids of the formula I see diagramm : EP0078362,P11,F3 in which R denotes hydrogen, methyl, ethyl or beta-hydroxyethyl, and their pharmaceutically usable acid addition salts and hydrates.
机译:1.索赔(针对缔约国:AT,BE,CH,DE,FR,GB,IT,LI,NL,SE)环丙基-6-氟-1,4-二氢-4-氧代-7-哌嗪子基-喹啉式I的-3-羧酸见图:EP0078362,P10,F3,其中R表示氢,甲基,乙基或β-羟乙基,及其药学上可用的酸加成盐,碱金属盐和水合物,但1-环丙基- 6-氟-1,4-二氢-4-氧-7-哌嗪基喹啉-3-羧酸及其盐酸盐1-环丙基-6-氟-1,4-二氢-4-氧-7-(4 -甲基哌嗪子基)-喹啉-3-羧酸和1-环丙基-6-氟-1,4-二氢-4-氧代-7-(4-乙基哌嗪子基)-喹啉-3-羧酸氢碘化物。 1.(对于缔约国LU而言)式I的1-环丙基-6-氟-1,4-二氢-4-氧代-7-哌嗪基-喹啉-3-羧酸的图式:EP0078362,P11,F3其中R表示氢,甲基,乙基或β-羟乙基,及其药学上可用的酸加成盐和水合物。

著录项

  • 公开/公告号JPH0244827B2

    专利类型

  • 公开/公告日1990-10-05

    原文格式PDF

  • 申请/专利权人 BAYER AG;

    申请/专利号JP19870127878

  • 申请日1987-05-25

  • 分类号A23K1/16;A23K1/17;A61K31/495;A61P31/04;C07C69/716;C07C69/738;C07D215/56;C07D401/00;

  • 国家 JP

  • 入库时间 2022-08-22 06:20:57

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