首页> 外国专利> AZELASTINE SALT, PREPARATION THEREOF, DRUG CONTAINING SAME AND HAVING ASTHMA-PREVENTIVE, ANTI-ALLERGIC, ANTIHISTAMINIC, ANTI-INFLAMMATORY, AND CEL-PROTECTIVE ACTION, AND PREPARATION OF SAID DRUG

AZELASTINE SALT, PREPARATION THEREOF, DRUG CONTAINING SAME AND HAVING ASTHMA-PREVENTIVE, ANTI-ALLERGIC, ANTIHISTAMINIC, ANTI-INFLAMMATORY, AND CEL-PROTECTIVE ACTION, AND PREPARATION OF SAID DRUG

机译:氮杂胺盐,其制备,含有相同且具有哮喘预防,抗过敏,抗组胺,抗炎和细胞保护作用的药物,以及所述药物的制备

摘要

The present invention relates to salts of azelastine having improved solubility in water. The salts of the present invention are prepared by reacting azelastine with acetic acid, gluconic acid, lactic acid, or malic acid. The azelastine salts are effective in providing a cytoprotective effect.
机译:本发明涉及在水中具有改善的溶解度的氮卓斯汀的盐。本发明的盐是通过使氮卓斯汀与乙酸,葡萄糖酸,乳酸或苹果酸反应制备的。氮卓斯汀盐可有效提供细胞保护作用。

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