首页> 外国专利> VERF. Z. PREPARATION OF A PYHSIC MIXTURE OF AT LEAST ONE SALT OF ((1-METHYL-1-PYRROLIDINIO) METHYL) -3-CEPHEM-4-CARBOXYLATE AND A PHARMACEUTICALLY CONFIDENT, NON-TOXIC, ORGANIC OR INORGANIC BASE

VERF. Z. PREPARATION OF A PYHSIC MIXTURE OF AT LEAST ONE SALT OF ((1-METHYL-1-PYRROLIDINIO) METHYL) -3-CEPHEM-4-CARBOXYLATE AND A PHARMACEUTICALLY CONFIDENT, NON-TOXIC, ORGANIC OR INORGANIC BASE

机译:VERF。 Z.制备至少(1-(1-甲基-1-吡咯烷基)甲基)-3-CEPHEM-4-羧酸酯盐和药学上机敏,无毒,有机或无机碱的羟基混合物

摘要

Temp. stable crystalline salts of alpha-(2-aminothiazol-4-yl) alpha-(Z)-methoxyiminoacetamido) -3 -(1-methyl-1-pyrrolidinio) methyl)-3-cephem-4-carboxylate (I) are claimed, selected from sulphuric, di-nitric, monohydrochloric and di-hydrochloric acid addn. salts and orthophosphoric acid addn. salts contg. 1.5-2 molar equivalents of H3PO4, or solvates of tehse. The salt may be mixed with a base e.g. L(+) lysine or L(+) arginine.
机译:温度要求保护α-(2-氨基噻唑-4-基)α-(Z)-甲氧基亚氨基乙酰氨基)-3-(1-甲基-1-吡咯烷基)甲基)-3-头孢-4-羧酸的稳定的结晶盐(I)选自硫酸,二硝酸,一盐酸和二盐酸。盐和正磷酸添加剂。盐续1.5-2摩尔当量的H3PO4或这些溶剂化物。可以将盐与碱例如碳酸氢钠混合。 L(+)赖氨酸或L(+)精氨酸。

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