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PROCESS FOR THE PREPARATION OF MEDICAL PRODUCTS CONTAINING AMINO-ACID DERIVATIVES AND PROCESS FOR THE PREPARATION OF MINO-ACID DERIVATIVES

机译:包含氨基酸衍生物的医药产品的制备方法和氨基酸衍生物的制备方法

摘要

Amino-acid derivatives of the formula I R1-CpH2p-(NH)q-CO-NH-CHR2-CO-Z-CmH2m-CHWR3-CO-NH-CHRSP 3-CR4-(CHR5)n- CO-E-Q-Y 1 in which R1 to R5, p, q, Z, m, n, E, Q, W and Y have the meanings given in Claim 1, and the salts thereof inhibit the activity of human plasma renin.
机译:式I的氨基酸衍生物R1-CpH2p-(NH)q-CO-NH-CHR 2 -CO-Z-CmH2m-CHWR <3> -CO-NH-CHR 3-CR <4 >-(CHR 5)n-CO-EQY 1,其中R 1至R 5,p,q,Z,m,n,E,Q,W和Y具有权利要求1中给出的含义及其盐抑制人血浆肾素的活性。

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