N-(HALOIDOPHENYL)-2-(BENZO-2,1,3-THIADIAZOL-4-SULPHONYL)AMINO-5-- CHLOROBENZAMIDES, SHOWING ACTIVITY IN EXPERIMENTAL TRICHOCEPHALIASIS

摘要

the invention u043eu0442u043du043eu0441u0438u0442u0441u00a0 to u0433u0435u0442u0435u0440u043eu0446u0438u043au043bu0438u0447u0435u0441u043au0438u043c u0441u043eu0435u0434u0438u043du0435u043du0438u00a0u043c, in particular to u0449u0433u0430u043bu043eu0438u0434 - u0444u0435u043du0438u043b) - 2 - {(u0431u0435u043du044du043e - 2,1,3 - u0442u0438u0430u0434u0438u0430u0437u043eu043b - 4 - u0441u0443u043bu044cu0444u043e neal) amino - 5 - u0445u043bu043eu0440u0431u0435u043du0437u0430u043cu0438u0434u0430u043c with u0430u043au0442u0438u0432u043d the pilot u0442u0440u0438u0445u043eu0446u0435u0444u0430u043bu0435u0437u0435 awn. objective u0432u044bu00a0u0432u043bu0435u043du0438u0435 more active compounds.synthesis of compounds by the reaction of 2 - {(benzo - 2,1,3 - u0442u0438u0430u0434u0438u0430u0437u043eu043b - 4 - u0441u0443u043bu044cu0444u043e neal) amino - 5 - u0445u043bu043eu0440u0431u0435u043du0437u043eu0439u043du043eu0439 acids with u0442u0438u043eu043du0438u043bu043eu043c and processing of u0445u043bu043eu0440u0430u043du0433u0438u0434u0440u0438u0434u0430 with 3.4 - u0434u0438u0445u043bu043eu0440u0430u043du0438u043bu0438u043du043eu043c or 4 - u0445u043bu043eu0440u0430u043du0438u043bu0438u043du043eu043c in u0434u0438u0445u043bu043eu0440u044du0442u0430u043du0435 in the presence of u0442u0440u0438u044du0442u0438u043bu0430u043cu0438u043du0430. exit%, u0442.u043fu043b., & deg; c; gross formula respectively, 72; 203 - 205; u044119u043du0446u04411u0437u043c u044eu043752, 65, 224, 226, CigHi2Cl2N 03S2... 1, table 2). (l, c