首页> 外国专利> PROCESS FOR PRODUCING ENDO-N-BRACES OPEN BRACKETS OPEN (8-METHYL-8-AZABICYCLO/3,2,1/OCTAN-3/YL)-AMINO BRACKETS CLOSED -CARBONYL BRACES CLOSED-2-(CYCLOPROPYLMETHOXY)-BENZAMIDE, ITS SALTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH COMPOUNDS AS ACTIVE INGREDIENT

PROCESS FOR PRODUCING ENDO-N-BRACES OPEN BRACKETS OPEN (8-METHYL-8-AZABICYCLO/3,2,1/OCTAN-3/YL)-AMINO BRACKETS CLOSED -CARBONYL BRACES CLOSED-2-(CYCLOPROPYLMETHOXY)-BENZAMIDE, ITS SALTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SUCH COMPOUNDS AS ACTIVE INGREDIENT

机译:制备ENDO-N括号的方法开环的化合物(8-甲基-8-氮杂双/ 3,2,1 / OCTAN-3 / YL)-氨基的化合物闭环-羰基的化合物闭环-2-(环丙基甲氧基)-苯甲酰胺包含此类化合物作为有效成分的盐和药物成分

摘要

(Endo)-N-[[(8-methyl-8-azabicyclo[3.2.1]octan-3-yl)amino]carbonyl]-2-( cyclop r opylmethoxy)benzamide and its pharmaceutically acceptable acid addition salts are useful as 5-HT3-antagonists, e.g. in the treatment of anxiety.
机译:(Endo)-N-[[((8-甲基-8-氮杂双环[3.2.1]辛烷-3-基)氨基]羰基] -2-(环磷酰甲氧基)苯甲酰胺及其药学上可接受的酸加成盐可用作5-HT3拮抗剂,例如在治疗焦虑症。

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