首页> 外国专利> MIXED PYRIDINE-2,4-AND-2,5-DICARBOXAMIDES, A PROCESS FOR PREPARING TEM, THE USE THEREOF AND PHARMACEUTICALS BASED ON THESE COMPOUNDS

MIXED PYRIDINE-2,4-AND-2,5-DICARBOXAMIDES, A PROCESS FOR PREPARING TEM, THE USE THEREOF AND PHARMACEUTICALS BASED ON THESE COMPOUNDS

机译:混合吡啶-2,4-和-2,5-二甲酰胺,一种制备TEM的方法,其使用和基于这些化合物的药物

摘要

The invention relates to mixed pyridine-2,4- and -2,5-dicarboxylic acid diamides, the carboxylic acid amide group in position 2 being a primary acid amide. The said compounds are suitable for the inhibition of proline hydroxylase and lysine hydroxylase and are used as fibrosuppressants and immunosuppressants.
机译:本发明涉及混合的吡啶-2,4-和-2,5-二羧酸二酰胺,第2位的羧酸酰胺基为伯酰胺。所述化合物适合于抑制脯氨酸羟化酶和赖氨酸羟化酶,并用作纤维抑制剂和免疫抑制剂。

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