首页> 外国专利> BIOERODIBLE IMPLANTABLE CONTROLLED RELEASE DOSAGE FORM COMPRISING A POLY(ORTHO ESTER) OR A POLYACETAL WITH AN ACTIVE AGENT INCORPORATED INTO THE CHAIN BACKBONE

BIOERODIBLE IMPLANTABLE CONTROLLED RELEASE DOSAGE FORM COMPRISING A POLY(ORTHO ESTER) OR A POLYACETAL WITH AN ACTIVE AGENT INCORPORATED INTO THE CHAIN BACKBONE

机译:包含链状骨中掺有活性剂的聚(Ortho酯)或聚脂的可生物降解的可控释放剂量形式

摘要

A bioerodible controlled release dosage form (1) is disclosed comprising a polymer formed by condensing beneficial agents (2) having a hydroxyl functionality of two or more with diketene acetals or divinyl ethers which delivers beneficial agents to a biological environment of use. A statistically significant portion of the beneficial agent (2) is covalently bonded within the polymer matrix (3). IMAGE
机译:公开了一种可生物蚀解的控释剂型(1),其包含通过将具有两个或多个羟基官能度的有益剂(2)与双烯酮缩醛或二乙烯基醚缩合而形成的聚合物,所述双烯酮缩醛或二乙烯基醚将有益剂递送至使用的生物环境。统计学上重要的有益剂(2)部分共价键合在聚合物基质(3)内。 <图像>

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