首页> 外国专利> NUCLEOSIDES, THEIR PREPARATION AND THEIR USE AS THERAPEUTIC AGENTS AND AS BUILDING BLOCKS OF SYNTHETIC OLIGONUCLEOTIDES

NUCLEOSIDES, THEIR PREPARATION AND THEIR USE AS THERAPEUTIC AGENTS AND AS BUILDING BLOCKS OF SYNTHETIC OLIGONUCLEOTIDES

机译:核苷,其制备及其作为治疗性寡核苷酸和合成寡核苷酸的构建基团的用途

摘要

New nucleosides having general formula (I), their preparation and their use are disclosed. These nucleosides show a therapeutic, in particular virostatic and cancerostatic action, and are very stable in comparison with analogous compounds. In addition, these compounds may be used as building blocks of synthetic oligonucleotides (ribo or 2'-desoxyribo forms).
机译:公开了具有通式(I)的新核苷,其制备和用途。这些核苷显示出治疗作用,特别是抗病毒和抗癌作用,并且与类似化合物相比非常稳定。另外,这些化合物可用作合成寡核苷酸(核糖或2'-脱氧核糖形式)的结构单元。

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