首页> 外国专利> THE USE OF COUMARINS AND 2-HYDROXYQUINOLINES AS PLA2 INHIBITORS, NOVEL COUMARINS AND 2-HYDROXYQUINOLINES, PROCESS OF THEIR PREPARATION AND MEDICAMENTS

THE USE OF COUMARINS AND 2-HYDROXYQUINOLINES AS PLA2 INHIBITORS, NOVEL COUMARINS AND 2-HYDROXYQUINOLINES, PROCESS OF THEIR PREPARATION AND MEDICAMENTS

机译:香豆素和2-羟基喹啉作为Pla2抑制剂,新型香豆素和2-羟基喹啉的用途,制备方法和药物

摘要

PCT No. PCT/EP94/02251 Sec. 371 Date Mar. 14, 1996 Sec. 102(e) Date Mar. 14, 1996 PCT Filed Jul. 9, 1994 PCT Pub. No. WO95/02588 PCT Pub. Date Jan. 26, 1995Use of compounds of formula I IMAGE (I) in which R1, R2, R3, R4, Y and Z have the meanings stated in the claims, tautomers thereof as well as their salts with non-toxic acids or bases for the production of pharmaceutical agents having an inhibitory action on PLA2 in addition to compounds of formula I in which X does not denote a valency and processes for the production thereof.
机译:PCT号PCT / EP94 / 02251第二部分371日期1996年3月14日102(e)日期1996年3月14日PCT 1994年7月9日提交PCT Pub。 WO95 / 02588 PCT公开号1995年1月26日日期R 1,R 2,R 3,R 4,Y和Z具有权利要求书中所述含义的式I (I)化合物及其互变异构体以及它们与无毒酸的盐的用途除了式I的化合物(其中X不表示化合价)以外,还生产用于对PLA2具有抑制作用的药物的碱及其制备方法。

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