17&bgr;-N-monosubstituted-carbamoyl-4-5&agr;-androst-1-en-3- ones of the formula ##STR1## wherein R.sup.1 is selected from hydrogen, methyl and ethyl and R.sup.2 is a branched chain alkyl of from 3-12 carbons, and R', R", R"' are hydrogen or methyl are active as testosterone 5&agr;- reductase inhibitors and thus are useful topically for treatment of androgenic alopecia.
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