首页> 外国专利> DERIVATIVES OF BETA-AMINO ACIDS SUBSTITUTED USEFUL AS INHIBITORS OF PLATELET AGGREGATION.

DERIVATIVES OF BETA-AMINO ACIDS SUBSTITUTED USEFUL AS INHIBITORS OF PLATELET AGGREGATION.

机译:有用的β-氨基氨基酸衍生物替代为血小板聚集的抑制剂。

摘要

NEW SUBSTITUTED AMINO-BETA ACID DERIVATIVES ARE PROVIDED THAT HAVE THE GENERAL FORMULA (AND) IN WHICH, FOR EXAMPLE, R2 IS SELECTED FROM THE GROUP WHICH CONSISTS OF HYDROGEN, RADICALS ALQUILY REDUCED, RADICALS ALQUINED, RADICALS ALQUINED, RADICALS ALQUINED, RADICALS ALQUINED, RADICALS ALQUINED ALICYCLIC, AROMATIC HYDROCARBON RADICALS, WHERE THE RADICALS ARE OPTIONALLY SUBSTITUTED WITH HYDROXY, ALCOXI REDUCED, ALKYL REDUCED, HALOGEN, NITRO, CIAN, AZIDO, UREID, CARBOXY, UREILENO, CARBON ARILSULFENIL, ALQUILSULFONIL, ARILSULFONIL, AMINO, ALQUILAMINO, TRIALQUILSILIL, AMINOSULFONIL, DIALQUILAMINO, ALCANOILAMINO, AROILAMINO, FENIL, REQUIRED, ALQUINIL, OQUIL, OQUIN AZIDA AND FENIL; THE INVENTION ALSO RELATES THE PHARMACEUTICAL COMPOSITIONS THAT INCLUDE SUCH DERIVATIVES.
机译:提供了新的取代的氨基二乙酸衍生物,其具有一般式(并且),例如,R 2从以下组中选择:氢,基团被减少,基团被确定,基团被确定,基团被确定自由基为脂环族,芳族烃基,其中自由基可选择性地被羟基,醇还原,烷基还原,卤素,硝基,茜素,氮杂环戊烯基,丙二烯基,醇,甲硅烷基,醇,甲硅烷基,脲,醇,甲硅烷基,脲,醇,甲硅烷基,脲,甲苯基氨基磺脲,二甲喹啉,阿尔卡诺胺,无芦荟素,茴香,必不可少的,喹诺酮,水,叠氮基和茴香;本发明还涉及包括这种衍生物的药物组合物。

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