首页> 外国专利> USE OF THIAZOLIDINE DERIVATIVES FOR PREPARING A PHARMACEUTICAL PREPARATION FOR TREATING IMPAIRED TOLERANCE OF GLUCOSE AND FOR PREVENTING OR DELAYING COMING OF DIABETES MELLITUS INDEPENDENTLY ON INSULIN

USE OF THIAZOLIDINE DERIVATIVES FOR PREPARING A PHARMACEUTICAL PREPARATION FOR TREATING IMPAIRED TOLERANCE OF GLUCOSE AND FOR PREVENTING OR DELAYING COMING OF DIABETES MELLITUS INDEPENDENTLY ON INSULIN

机译:噻唑烷衍生物的用途用于制备药物制剂以治疗糖耐量降低以及预防或延缓糖尿病在糖尿病患者中的发作

摘要

The use of a compound of formula (IX) or a tautomeric form thereof and / or a pharmaceutically acceptable salt thereof and / or a pharmaceutically acceptable solvate thereof, wherein A.sub.5. means a substituted or unsubstituted aromatic heterocyclic group, A.sub.6.n. means a benzene ring having up to a total of 5 substituents, X.sub.6. means an oxygen, sulfur or NR.sub.3n group in which R.sub.32.n. means a hydrogen atom, an alkyl group, an acyl group or an aralkyl group in which the aryl moiety may be substituted or unsubstituted, or a substituted or unsubstituted aryl group, Y.sub.2. means an oxygen or sulfur atom, R.sub.31.n. is a hydrogen atom or an alkyl group, an aralkyl group or an aryl group, and n is a number from 2 to 6, for the manufacture of a medicament preparation or treatment of impaired glucose tolerance to prevent or delay the onset of insulin-independent diabetes mellitus.ŕ
机译:式(IX)的化合物或其互变异构形式和/或其药学上可接受的盐和/或其药学上可接受的溶剂化物的用途,其中A.sub.5。 ″取代的或未取代的芳族杂环基,A.sub.n。″。术语“苯环”是指具有最多5个取代基X 6的苯环。表示氧,硫或NR 3n基团,其中R 32 n。术语“芳基”是指氢原子,烷基,酰基或芳烷基,其中芳基部分可以被取代或未被取代,或被取代或未被取代的芳基Y.sub.2。 R 31是指氧或硫原子。 n是氢原子或烷基,芳烷基或芳基,并且n是2至6的数字,用于制造药物制剂或治疗葡萄糖耐量降低,以预防或延迟胰岛素非依赖性发作糖尿病。ŕ

著录项

  • 公开/公告号CZ283208B6

    专利类型

  • 公开/公告日1998-01-14

    原文格式PDF

  • 申请/专利权人 SANKYO COMPANY;

    申请/专利号CZ19960002823

  • 申请日1994-09-14

  • 分类号A61K31/41;A61K31/42;A61K31/425;A61K31/44;A61K31/495;A61K31/505;

  • 国家 CZ

  • 入库时间 2022-08-22 02:58:24

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号