首页> 外国专利> PREPARATION OF 5-2-ETHOXY-5-(4-METHYLPIPERAZIN-1-YLSULPHONYL)PHENYL-1-METHYL -3-(N-PROPYL)-1,6-DIHYDRO-7H-PYRAZOLO4,3-DPYRIMIDIN-7-ONE(SIL DENAFIL) AND INTERMEDIATES DENA 5-2-ETHOXY-5-(4-METHYLPIPERAZIN-1-YLSULPHONYL)PHENYL-1-METHYL -3-(N- PROPYL)-1,6-DIHYDRO-7H-PYRAZOLO4,3-DPYRIMIDIN-7-ONE(SLIDENAFI L);INT ERMEDIATES

PREPARATION OF 5-2-ETHOXY-5-(4-METHYLPIPERAZIN-1-YLSULPHONYL)PHENYL-1-METHYL -3-(N-PROPYL)-1,6-DIHYDRO-7H-PYRAZOLO4,3-DPYRIMIDIN-7-ONE(SIL DENAFIL) AND INTERMEDIATES DENA 5-2-ETHOXY-5-(4-METHYLPIPERAZIN-1-YLSULPHONYL)PHENYL-1-METHYL -3-(N- PROPYL)-1,6-DIHYDRO-7H-PYRAZOLO4,3-DPYRIMIDIN-7-ONE(SLIDENAFI L);INT ERMEDIATES

机译:制备5- [2-乙氧基-5-(4-甲基哌嗪-1-甲苯基)苯基] -1-甲基-3-(正丙基)-1,6-二羟基-7H-吡唑并[4,3-D ] PYRIMIDIN-7-ONE(SIL DENAFIL)并中间体DENA 5- [2-ETHOXY-5-(4-METHYLPIPERAZIN-1-YLSULPHONYL)PHENYL] -1-METHYL-3--3-(N-PROPYL)-1,6- DIHYDRO-7H-PYRAZOLO [4,3-D] PYRIMIDIN-7-ONE(SLIDENAFI L); INT中介

摘要

A process for the preparation of a compound of formula (I): CHEM also knows as sildenafil which comprises cyclisation of a compound of formula (II): CHEM
机译:制备式(I):的化合物的方法,也称为西地那非,其包括环化式(II)的化合物:

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