DERIVATIVES OF BENZOXACINA, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICS.

摘要

COMPOUND RESPONDING TO THE GENERAL FORMULA (I) IN WHICH AND REPRESENTS AN ATOM OF HYDROGEN, FLUORINE OR CHLORINE OR A METHYL OR METOXI GROUP, REPRESENTING R1 WELL A PHENYLUS GROUP REPLACED BY AN ATHLE OF FLUORIDE OR BY A SELECTED GROUP THE METHYL, METOXI, TRIFLUORMETHYL AND PHENYLUS GROUPS, OR A TEN-2YL GROUP, REPRESENTING R2 A METHYL GROUP, R3 REPRESENTING A (C1-C4) GROUP ALKYLALLY ALSO, A SUITABLE ALKILE EVENT NUCLEUS FOR 2 TO 3 METOXI GROUPS, WELL A GROUP 2- (PIRIDIN-2-IL) ETHYL, OR R2 AND R3 FORMAN, WITH NITROGEN, WELL A 4-PHENYL GROUP (PIPERIDIN-1-ILO), WELL A GROUP 4-PHENYLMETHYLL (PIPERIDIN-1-ILO), WELL A GROUP 1,2,3,4TETRAHIDROISOQUINOLEIN-2-ILO, WELL A GROUP 6-METOXI-1,2,3,4TETRAHYDROISOIQUINOLEIN-2YL, WELL A GROUP 5,8, DIMETOXI-1,2,3,4TETRAHIDROISOQUINOLEIN-2-ILO, WELL A GROUP 6,7-DIMETOXI-1,2,3,4TETRAHIDROISOQUINOLEIN-2-ILO, WELL A GROUP 2,3,4,5-TETRAHIDRO1H-3 - BENZACEPIN-3-ILO, WELL A GROUP 7,8-DIMETOXI-2,3,4,5TETRAHIDRO 1H-3-BENZACEPIN-3-ILO, AND X REPRESENTS A CARBONYL GROUP WELL, A SULPHONYL GROUP WELL. APPLICATION IN THERAPY.