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N-METHYL-D-ASPARTATE RECEPTOR CHANNEL BLOCKERS AND METHOD FOR IDENTIFYING SUCH

机译:N-甲基-D-天冬氨酸受体通道阻滞剂和鉴定这种物质的方法

摘要

Compounds that provide protection against excitotoxic neuronal damage are selected from the group consisting of Arg-rich oligopeptides and compounds of formula (1), where R1 is alkyl, alkenyl, or hydroxyalkyl, aminoalkyl, or alkoxy-alkyl; and R2 and R3 are each natural or artificial amino acid side chains.
机译:提供保护免受兴奋性神经元损伤的化合物选自富含Arg的寡肽和式(1)的化合物,其中R 1为烷基,烯基或羟烷基,氨基烷基或烷氧基-烷基; R2和R3分别是天然或人工氨基酸侧链。

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