首页> 外国专利> AMINO-SUBSTITUTED THIADIAZOLES, PYRIMIDINES, TRIAZINES OR TRIAZOLES USEFUL AS CTF RECEPTOR ANTAGONISTS

AMINO-SUBSTITUTED THIADIAZOLES, PYRIMIDINES, TRIAZINES OR TRIAZOLES USEFUL AS CTF RECEPTOR ANTAGONISTS

机译:氨基取代的噻唑类,嘧啶类,三嗪类或三唑类,可用作CTF受体拮抗剂

摘要

CRF receptor antagonists are disclosed. Such receptor antagonists are thiadiazole-, pyrimidine-, triazine-, and triazole-containing compounds substituted with both a C3-C14 monocyclic or fused, homoaryl or heteroaryl group and a substituted amine group. The CFR receptor antagonists have utility in the treatment of a variety of disorders, including disorders associated with the hypersecretion of CRF.
机译:公开了CRF受体拮抗剂。这样的受体拮抗剂是被C 3 -C 14单环或稠合的均芳基或杂芳基和取代的胺基取代的含噻二唑,嘧啶,三嗪和三唑的化合物。 CFR受体拮抗剂可用于治疗多种疾病,包括与CRF过度分泌有关的疾病。

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