首页> 外国专利> (2R, 3S) DIHYDRATE -3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY- 3-PHENYLPROPIONATE OF 4,10BETA-DIACETOXY-2ALPHA-BENZOYLOXY- 5BETA, 2O-EPOXY-1-HYDROX CYCLOPROPA (G) TAX-11- ENE-13ALPHA-YLE, AND PREPARATION METHOD THEREOF

(2R, 3S) DIHYDRATE -3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY- 3-PHENYLPROPIONATE OF 4,10BETA-DIACETOXY-2ALPHA-BENZOYLOXY- 5BETA, 2O-EPOXY-1-HYDROX CYCLOPROPA (G) TAX-11- ENE-13ALPHA-YLE, AND PREPARATION METHOD THEREOF

机译:(2R,3S)(3-R)3-叔丁基羰基氨基-2-羟基-4,10BETA-二乙酰氧基-2ALPHA-苯氧基-5BETA,2O-环氧-1-羟基环丙酸酯(G)税11-ENE-的3-苯基丙酸酯13α-紫杉醇及其制备方法

摘要

A 4,10 beta -diacetoxy-2 alpha -benzoyloxy-5 beta ,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa[g]tax-11-ene-13 alpha -yl (2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate, and the preparation thereof by crystallisation from a water-alcohol or water-ketone solution, are disclosed.
机译:4,10β-二乙酰氧基-2α-苯甲酰氧基-5β,20-环氧-1-羟基-9-氧代-19-正环丙烷[g] tax-11-ene-13α-基(2R,3S公开了)-3-叔丁氧基羰基氨基-2-羟基-3-苯基丙酸酯二水合物,以及通过从水-醇或水-酮溶液中结晶而制备的方法。

著录项

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号