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Compounds which are derivatives of imidazobenzoxazine, 1995 of preparation and their uses in international application no.
Compounds which are derivatives of imidazobenzoxazine, 1995 of preparation and their uses in international application no.
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机译：作为咪唑并苯并恶嗪衍生物的化合物，1995年制备及其在国际申请No.
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摘要
Imidazo benzoxazine derivatives of formula (I), their pure and mixed enantiomers, including racemic mixtures and acid addition salts are new. R1, R2 = H, alkyl, alkenyl, cycloalkyl, cycloalkenyl, or alkylene-cycloalkyl; or R1+R2 = cycloalkyl; R3 = H, halo, nitro, amino, alkylamino, dialkylamino, acylamino, cyano, carboxamide, -COOH, amino-methylene, amidino, alkyl, fluoroalkyl, aralkylamino, -SO2NR5R6 or -NR7SO2R8; R5-R8 = H or alkyl; R4 = H, alkyl, alkenyl, cycloalkyl, cycloalkenyl, aralkyl, alkoxyalkyl, fluoroalkyl, phenoxyalkyl, -(CH2)m-NR9SO2R10, -(CH2)z-SO2NR11R12 or -(CH2)v-CONR13R14; m, v, z = 2 or 3; R9-R14 = H, alkyl, alkenyl, cycloalkyl or cycloalkenyl; Y = O, NH, N-alkyl or S; n = 0-2.
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机译：式（I）的咪唑并苯并恶嗪衍生物，其纯的和混合的对映异构体，包括外消旋混合物和酸加成盐是新的。 R1，R2 ＝ H，烷基，烯基，环烷基，环烯基或亚烷基-环烷基;或R 1 + R 2 ＝环烷基;或R3 = H，卤素，硝基，氨基，烷基氨基，二烷基氨基，酰基氨基，氰基，羧酰胺，-COOH，氨基-亚甲基，a基，烷基，氟代烷基，芳烷基氨基，-SO2NR5R6或-NR7SO2R8; R5-R8 ＝ H或烷基; R4 = H，烷基，烯基，环烷基，环烯基，芳烷基，烷氧基烷基，氟代烷基，苯氧基烷基，-（CH2）m-NR9SO2R10，-（CH2）z-SO2NR11R12或-（CH2）v-CONR13R14; m，v，z = 2或3; R9-R14 ＝ H，烷基，烯基，环烷基或环烯基; Y ＝ O，NH，N-烷基或S; n = 0-2。
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