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PREPARATION FOR SUSTAINED RELEASE OF DICLOFENAC SODIUM

机译:持续释放双氯芬酸钠的制备

摘要

PROBLEM TO BE SOLVED: To obtain a preparation of diclofenac sodium, easily produced, and excellent in sustained release of diclofenac sodium and in its preservation stability. ;SOLUTION: This preparation for sustained release of diclofenac sodium is obtained by coating a core granule containing diclofenac sodium and phosphoric acid or its salt as the acidic component with a film for sustained release, which is made of a mixture of a hydroxypropylmethyl cellulose acetate and aminoalkyl methacrylate-based copolymer in a weight ratio of (3:7) to (8:2).;COPYRIGHT: (C)1999,JPO
机译:解决的问题:获得易于制备的双氯芬酸钠的制剂,该制剂在双氯芬酸钠的持续释放和保存稳定性方面极好。 ;解决方案:这种双氯芬酸钠持续释放的制剂是通过在由双氯芬酸钠和磷酸或其盐作为酸性成分的核心颗粒上涂覆一层持续释放的薄膜制成的,该薄膜由羟丙基甲基乙酸纤维素和重量比为(3:7)与(8:2)的基于甲基丙烯酸氨基烷基酯的共聚物。;版权:(C)1999,JPO

著录项

  • 公开/公告号JPH1160477A

    专利类型

  • 公开/公告日1999-03-02

    原文格式PDF

  • 申请/专利权人 MAEDA YAKUHIN KOGYO KK;

    申请/专利号JP19970230237

  • 发明设计人 KOYAMA HARUKI;OOUCHI MASATO;

    申请日1997-08-12

  • 分类号A61K31/19;A61K9/52;A61K47/30;

  • 国家 JP

  • 入库时间 2022-08-22 02:32:32

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