首页> 外国专利> NEW ANDROSTA-1,4-DIENE OR-1,3,5-TRIENE DERIVATIVES AS INTERMEDIATES FOR 6-ALPHA,9-ALPHA-DIFLUORIZED-STEROIDES

NEW ANDROSTA-1,4-DIENE OR-1,3,5-TRIENE DERIVATIVES AS INTERMEDIATES FOR 6-ALPHA,9-ALPHA-DIFLUORIZED-STEROIDES

机译:新的ANDROSTA-1,4-二烯OR-1,3,5-三烯衍生物作为6-α,9-α-二恶英的中间体

摘要

the invention is a new u00e1ltalu00e1nu0151s formula (vi) andru0151szta - 1,4 - diene - or - 1,3,5 - triu00e9n - in the formula, r szu00e1rmazu00e9ku0151kra hidru0151gu00e9natu0151m vagyu00e9sztermaradu00e9k report, report hidru0151gu00e9n x - or flu0171u0151ratu0151m,the pu0151ntu0151zu0151ttvu0151nalakkal y y, together with 3 - - - a system that u0151xu0151 d4, or x and y jelentu00e9sehidru0151gu00e9natu0151m, together with the pu0151ntu0151zu0151tt vu0151nalakkal or1 - 3 - d - 3,5 - rendszertjelent,the report ahu0151l u0171tu00f3bbinu00e1l r1 enu0151l ether or enu0151l - u00e9sztermaradu00e9ka, vu0151natku0151zik.these can be used in the known gyu0171lladu00e1sgu00e1tlu00f3hatu00e1su00fa, (i) u00e1ltalu00e1nu0151s 6a, 9a - diflu0171u0151ru0151zu0151tt zteru0151idu0151k (ii) compounds of the formula kiindu0171lva, u0151xidu00e1lu00f3lebu0151ntu00e1s,the 6 - helyzetbenflu0171u0151ru0151zu00e1s and, finally, the epu0151xid, by means of a flu0171u0151rhidratu00e1lu00e1sa.
机译:本发明是新的公式(vi)并且公式中的r u0151szta-1,4-二烯-或-1,3,5-tri u00e9n-r sz u00e1rmaz u00e9k u0151kra hidr u0151g u00e9nat u0151m vagy u00e9sztermarad u00e9k报告,报告hidr u0151g u00e9n x-或fl u0171 u0151rat u0151m,p u0151nt u0151z u0151ttv和u015ynal-- u0151x u0151 d4或x和y jelent u00e9sehidr u0151g u00e9nat u0151m,以及p u0151nt u0151z u0151tt v u0151nalakkal或1-3-d-3,5-rendszertahlent, u0151l u0171t u00f3bbin u00e1l r1 en u0151l以太或en u0151l- u00e9sztermarad u00e9ka,v u0151natk u0151zik。这些可用于已知的gy u0171llad u00e1sg u00e1sg i) u00e1ltal u00e1n u0151s 6a,9a-difl u0171 u0151r u0151z u0151tt zter u0151id u0151k(ii)式kiind u0171lva, u0151xid u00e1l u00f3leb u00u1nt -helyzetbenfl u0171 u0151r u0151z u00e1s,最后是ep u015 1xid,通过fl u0171 u0151rhidrat u00e1l u00e1sa。

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