首页> 外国专利> PROCESS FOR PRODUCING 1-SUBSTITUTED ARYL-1,4-DIHYDRO-4-OXONAPHTHYRIDINE DERIVATIVE, INTERMEDIATES THEREFOR AND PROCESSES FOR PRODUCING THE INTERMEDIATES

PROCESS FOR PRODUCING 1-SUBSTITUTED ARYL-1,4-DIHYDRO-4-OXONAPHTHYRIDINE DERIVATIVE, INTERMEDIATES THEREFOR AND PROCESSES FOR PRODUCING THE INTERMEDIATES

机译:生产1-取代的芳基-1,4-二氢-4-氧杂吡啶吡啶衍生物的中间体,中间体和中间体的制备方法

摘要

This invention relates to a process for industriallyproducing a 11-substituted aryl-1,4-dihydro-oxonaphthyridinederivative and a salt thereofwherein R1 represents a hydrogen atom or a carboxyl-protectinggroup; R2a represents a 3-amino-1-pyrrolidinyl group in which theamino group may be protected, or a 1-piperazinyl group in whichthe imino group may be protected; and X represents a hydrogenatom or a fluorine atom, which are useful as an antibacterialagent, and also to intermediates therefor and processes forproducing the intermediates.
机译:本发明涉及工业上的方法产生11-取代的芳基-1,4-二氢-氧代萘啶衍生物及其盐其中R1代表氢原子或羧基保护基组; R 2a代表3-氨基-1-吡咯烷基,其中氨基可以被保护,或者其中的1-哌嗪基可以被保护亚氨基可能受到保护; X代表氢原子或氟原子,可用作抗菌剂剂及其中间体和方法生产中间体。

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