首页>
外国专利>
METHOD OF TREATMENT OR PROPHYLAXIS OF MAMMALS AND HUMAN WITH VOMITING USING SOME QUINUCLIDINE, PIPERIDINE, AZANORBORNANE, ETHYLENEDIAMINE DERIVATIVES AND RELATED COMPOUNDS
METHOD OF TREATMENT OR PROPHYLAXIS OF MAMMALS AND HUMAN WITH VOMITING USING SOME QUINUCLIDINE, PIPERIDINE, AZANORBORNANE, ETHYLENEDIAMINE DERIVATIVES AND RELATED COMPOUNDS
FIELD: organic chemistry, pharmacology. SUBSTANCE: method involves treatment or prophylaxis of mammals with vomiting using the following compounds: (2S, 3S)-N-(5-tert. -butyl-2-methoxy- -phenyl)-methyl-2-diphenylmethyl-1-azadicyclo(2,2,2)octane-3- -amine, (2S,3S)-N-(5-isopropyl-2-methoxyphenyl)-methyl-2- -diphenylmethyl-1-azadicyclo(2,2,2)octane-3-amine and (2S, 3S)-2-phenyl-3-(2-methoxy-5-trifluoromethoxybenzyl)- -aminopiperidine. EFFECT: enhanced effectiveness of treatment. 3 cl, 24 dwg, 3 ex
展开▼
机译:领域:有机化学,药理学。物质:该方法涉及使用以下化合物进行呕吐的哺乳动物的治疗或预防:(2S,3S)-N-(5-叔丁基-丁基-2-甲氧基-苯基)-甲基-2-二苯基甲基-1-氮杂二环( 2,2,2)辛烷-3-胺,(2S,3S)-N-(5-异丙基-2-甲氧基苯基)-甲基-2--二苯甲基-1-氮杂二环(2,2,2)辛烷- 3-胺和(2S,3S)-2-苯基-3-(2-甲氧基-5-三氟甲氧基苄基)-氨基哌啶。效果:增强治疗效果。 3 cl,24 dwg,3 ex
展开▼