首页> 外国专利> HETEROCYCLIC COMPOUNDS AND COMPOSITION ON SAID SHOWING ANTAGONISTIC EFFECT WITH RESPECT TO TACHYKININ RECEPTORS

HETEROCYCLIC COMPOUNDS AND COMPOSITION ON SAID SHOWING ANTAGONISTIC EFFECT WITH RESPECT TO TACHYKININ RECEPTORS

机译:杂环化合物及其与速激肽受体相关的显示抗拮抗作用的成分

摘要

Compounds of formula (I): CHEM and the quaternary ammonium derivatives thereof, especially compounds in which L represents a group CHEM have tachykinin receptor antagonist activity and exhibit an activity against both the NK1 receptors and the NK2 receptors.
机译:式(I)的化合物:及其季铵衍生物,特别是其中L代表基团的化合物具有速激肽受体拮抗剂活性,并且对NK1受体和NK2受体均具有活性。

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