首页> 外国专利> PHYSICALLY STABLE AND X-RAY AMORPHOUS FORM OF HYDROCHLORIDE RANITIDINE HAVING AN INCREASED ANTI-ULCER ACTIVITY AND METHOD FOR PRODUCING THE SAME

PHYSICALLY STABLE AND X-RAY AMORPHOUS FORM OF HYDROCHLORIDE RANITIDINE HAVING AN INCREASED ANTI-ULCER ACTIVITY AND METHOD FOR PRODUCING THE SAME

机译:具有增强的抗溃疡活性的盐酸拉尼替丁的物理稳定和X射线非晶体形式及其制备方法

摘要

The present invention relates to a new and formerly known form of hydrochloride ranitidine having H2-blocking properties. This form is X-ray amorphous, substantially differs from the formerly known crystalline modifications due to its characteristics, and also exhibits an enhanced anti-ulcer effect. This X-ray amorphous form is physically stable and can be used in medicine. This invention also relates to a method for producing this X-ray amorphous form from formerly known crystalline modifications.
机译:本发明涉及具有H 2阻断性质的盐酸盐雷尼替丁的新的和先前已知的形式。该形式是X射线无定形的,由于其特性而与先前已知的晶体修饰显着不同,并且还表现出增强的抗溃疡作用。这种X射线无定形形式在物理上稳定,可用于医学。本发明还涉及由先前已知的结晶变体生产该X射线无定形形式的方法。

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