首页> 外国专利> New 2-heteroaryl-5-phenyl-3,4-dihydro-2H-pyrrole derivatives, useful as insecticides, acaricides or nematocides, e.g. for protection of plants or wood, or as veterinary ectoparasiticides

New 2-heteroaryl-5-phenyl-3,4-dihydro-2H-pyrrole derivatives, useful as insecticides, acaricides or nematocides, e.g. for protection of plants or wood, or as veterinary ectoparasiticides

机译:新的2-杂芳基-5-苯基-3,4-二氢-2H-吡咯衍生物,可用作杀虫剂,杀螨剂或杀线虫剂,例如用于保护植物或木材,或用作兽用抗寄生虫药

摘要

2-Heteroaryl-5-phenyl-3,4-dihydro-2H-pyrrole derivatives (I) are new. Pyrroline derivatives of formula (I) are new: Het = optionally substituted (os), unsaturated 5-10 membered mono- or bicyclic heterocycle (e.g. 5- or 6-membered monocyclic heterocycle containing one or more of N, O and S); m = 0-4; R1 = halo, -X-A, -B-Z-D or -Y-E; R2 = H, halo, CN, NO2, alkyl, alkoxy, haloalkyl, haloalkoxy, alkoxyalkoxy or S(O)oR3; o = 0-2; R3 = alkyl or haloalkyl; X = direct bond, O, S, CO, COO, OCO, alkylene, alkenylene, alkynylene, oxyalkylene, thioalkylene, alkylenedioxy or dialkylsilylene; A = phenyl, naphthyl, tetrahydronaphthyl or 5-10 membered heterocycle containing 1 or 2 aromatic rings and one or more of O, S and N (all os); B = os p-phenylene; Z = O or S; D = H, alkyl, alkenyl, alkynyl, haloalkyl or haloalkenyl; or cycloalkyl, cycloalkylalkyl, cycloalkenyl, cycloalkenylalkyl, phenylalkyl, naphthylalkyl, tetrahydronaphthyl-alkyl or heteroarylalkyl (all os); or -COR4, -CONR5R6 or -(CH2)p-CR7R8)q-(CH2)r-G; or -Z-D = os phenoxyalkyl; Y = direct bond, O, S, CO, COO, OCO, alkylene, alkenylene, alkynylene, alkyleneoxy, oxyalkylene, thioalkylene, alkylenedioxy or as for B; E = H, alkyl, alkenyl, alkynyl, haloalkyl or haloalkenyl; cycloalkyl, cycloalkenyl, phenyl or heteroarylalkyl (all os); or -(CH2)p-CR7R8)q-(CH2)r-G; R4 = alkyl, alkoxy, alkenyl or alkenyloxy; or cycloalkyl, cycloalkoxy, cycloalkylalkoxy, phenyl or naphthyl (all os); R5, R7, R8 = H or alkyl; R6 = alkyl or haloalkyl; or cycloalkyl, cycloalkylalkyl, phenyl or phenylalkyl (all os); p, q, r = 0-3, provided that their sum is less than 6; G = CN; os 5- or 6-membered heterocycle; or a wide range of other substituents. An Independent claim is included for the preparation of (I). Full Definitions are given in the 'DEFINITIONS - Preferred Definitions' field.
机译:2-杂芳基-5-苯基-3,4-二氢-2H-吡咯衍生物(I)是新的。式(I)的吡咯啉衍生物是新的:Het =任选取代的(os),不饱和的5-10元单环或双环杂环(例如含有N,O和S中的一个或多个的5元或6元单环杂环); m = 0-4; R1 =卤素,-X-A,-B-Z-D或-Y-E; R2 = H,卤素,CN,NO2,烷基,烷氧基,卤代烷基,卤代烷氧基,烷氧基烷氧基或S(O)oR3; o = 0-2; R3 =烷基或卤代烷基; X =直接键,O,S,CO,COO,OCO,亚烷基,亚烯基,亚炔基,氧亚烷基,硫代亚烷基,亚烷基二氧基或二烷基亚甲硅烷基; A =苯基,萘基,四氢萘基或5-10元杂环,其含有1或2个芳环和一个或多个O,S和N(全部为os); B =邻对亚苯基; Z = O或S; D = H,烷基,烯基,炔基,卤代烷基或卤代烯基;或环烷基,环烷基烷基,环烯基,环烯基烷基,苯烷基,萘基烷基,四氢萘基烷基或杂芳基烷基(全部为os);或或-COR4,-CONR5R6或-(CH2)p-CR7R8)q-(CH2)r-G;或-Z-D = os苯氧基烷基;或Y =直接键,O,S,CO,COO,OCO,亚烷基,亚烯基,亚炔基,亚烷氧基,氧亚烷基,硫代亚烷基,亚烷基二氧基或对于B而言; E = H,烷基,烯基,炔基,卤代烷基或卤代烯基;环烷基,环烯基,苯基或杂芳基烷基(全部为os);或-(CH2)p-CR7R8)q-(CH2)r-G; R4 =烷基,烷氧基,烯基或烯氧基;或环烷基,环烷氧基,环烷基烷氧基,苯基或萘基(全部为os);或R5,R7,R8 = H或烷基; R6 =烷基或卤代烷基;或环烷基,环烷基烷基,苯基或苯烷基(全为os);或p,q,r = 0-3,条件是它们的总和小于6; G = CN; os 5或6元杂环;或各种各样的其他取代基。准备(I)包括独立权利要求。完整定义在“定义-首选定义”字段中给出。

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