HETEROCYCLIC BENZOYL-GUANIDINE DERIVATIVES SUBSTITUTED WITH N-OXIDE, PROCESS FOR PRODUCING THEM, THEIR USE FOR PRODUCING PHARMACEUTICALS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

摘要

In the compounds of the invention (I), R (1) is trifluoromethyl, halogen or -SOu-R (22) wherein u is 1 or 2, R (22) is alkyl of 1 to 7 carbon atoms, R (2) is Hetoxy, where Het is N-oxide of pyridyl or quinolyl optionally substituted with 1-3 methyl, R (3), R (4) and R (5) being hydrogen. The invention relates to the preparation of the above compounds and their use as a medicament or diagnostic agent. ŕ